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瑞禧定制抗体偶联药物Auristatin F/HTI-286/TubulysinM/Maytansinoid AP-3/DM1/DM

时间:2021-04-29 16:39:47       浏览:525

Auristatin F是细胞毒性分子,微管蛋白修饰分子,强效抗**活性,MMAF的类似物以及在抗体药物偶连体开发中作为毒素分子。

 英文名称:Auristatin F

中文名称:奥瑞他汀 F

CAS:163768-50-1




抗体药物偶联物(Antibody-drug conjugate, ADC)是通过化学键将具有生物活性的细胞毒药物连接到单克隆抗体(mAb)上,单克隆抗体(mAb)作为载体将细胞毒药物靶向运输到目标细胞中发挥作用的一类药物。既具有细胞毒药物杀伤力强大的特点,又结合了重组单克隆抗体(mAb)高度的靶向性,稳定性和有利的药代动力学特征,主要表现为:治疗效力强;特异性高;免疫原性弱,不容易产生抗药性;血清中循环时间长(短于单抗);对非靶点毒性弱等。

 

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OSu-Glu-vc-PAB-MMAE

SMCC-DM1

SPDB-DM4

OSu-PEG4-vc-PAB-DMEA
Duocarmycin SA

Mylotarg-linker

OSu-Glu-vc-PAB-MMAD

Sulfo-SPDB-DM4

IMGN779-linker

OSu-PEG4-vc-PAB-DMEA

Duocarmycin TM

OSu-PEG4-vc-PAB-DMEA
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MC-vc-PAB-MMAE

MC-MMAF

MC-DM1

MC-MMD-10

MA-PEG4-vc-PAB-DMEA-duocarmycin SA

MC-vc-PAB-C6-a-amanitin

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MC-vc-PAB-DMEA-(PEG2)-duocarmycin SA

MC-vc-PAB-Tubulysin M

MC-va-PAB-MMAD

MA-PEG4-VC-PAB-DMAE-PNU159682

MA-PEG4-VA-PBD

MC-vc-PAB-MMAF

MC-vc-PAB-MMAD

MC-vc-PAB-Auristatin 0101

MA-PEG8-VA-PAB-SG3199

CL2A-SN 38

MC-GGFG-DX8951

MEDI4276_linker payload

MA-PEG4-vc-PAB-DMEA-duocarmycin TM

MC-vc-PAB-(PEG2)-duocarmycin TM

MA-PEG4-vc-PAB-DMEA-duocarmycin DM

MC-vc-PAB-(PEG2)-duocarmycin DM

DGN549

MPB-vc-PAB-MMAE

MPB-MMAF

DBCO-PEG4-vc-PAB-MMAE

DBCO-PEG4-MMAF

DBCO-PEG4-Ahx-DM1

DBCO-PEG4-vc-PAB-Duocarmycin SA

DBCO-PEG4-vc-PAB-(PEG2)-Duocarmycin SA

DBCO-PEG4-VA-PBD

DBCO-PEG4-vc-PAB-MMAF

DBCO-PEG4-vc-PAB-MMAD

DBCO-PEG4-vc-PAB-Duocarmycin TM

DBCO-PEG4-vc-PAB-(PEG2)-Duocarmycin TM

DBCO-PEG4-vc-PAB-Duocarmycin DM

DBCO-PEG4-vc-PAB-(PEG2)-Duocarmycin DM

DBCO-PEG4-VC-PAB-DMAE-PNU159682

DBCO-PEG4-DMAE-PNU159682

DBCO-PEG4-GGFG-DX8951

DBCO-PEG4-vc-PAB-Ahx-DM1

DBCO-PEG8-VA-PAB-SG3199

Gly3-vc-PAB-MMAE

Gly3-MMAF

Gly5-Ahx-DM1

PNU159682-EDA-Gly3

ADC pre-screening kit A

Protein A-DM1

Protein A-MMAE

Protein A-MMAF

Protein A-Duocarmycin

Protein A-Calicheamicin

Protein A-PBD

ADC pre-screening kit G

Protein G-DM1

Protein G-MMAE

Protein G-MMAF

Protein G-Duocarmycin

Protein G-Amanitin

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Rabbit Anti-vc-PAB-MMAE pAb

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Mouse Anti-MMAF mAb (F3B11)

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Mouse Anti-MMAE /F mAb (C12A1)

Rabbit Anti-DM1/4 pAb

Mouse Anti-DM1/4 mAb (F1D5)

Mouse Anti-DM1/4 mAb (G2F3)

Rabbit Anti-Calicheamicin pAb

Mouse Anti-Calicheamicin mAb (B1G9)&

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