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Biotin-雷公藤甲素,生物素修饰雷公藤甲素
| Catalog # | Pkg Size | Price | Quantity | Shopping Cart |
|---|---|---|---|---|
| R-667 | 10mg | ¥ 4800 | 加入购物车 | |
结构式
| 外观 | N/A |
| 分子量 | N/A |
| 溶解度 | N/A |
| CAS号 | N/A |
| 质量控制 | N/A |
| 储存条件 | N/A |
| 保存时间 | N/A |
| 其他信息 | N/A |
生物素修饰雷公藤甲素完整保留环氧内酯活性骨架,不破坏原药靶向结合能力,是中药单体靶点筛选探针。分子可跨膜进入细胞,与胞内作用蛋白特异性结合,后续经链霉亲和素磁珠富集复合物,质谱鉴定结合靶点,解析雷公藤甲素免疫抑制、抗肿瘤分子机制。脂溶性探针,母液采用 DMSO 配制,生理缓冲液稀释给药细胞。常用于免疫药理研究、天然产物靶点发掘、先导化合物作用机制验证,需低温避光密闭储存,规避高温与酸碱造成内酯环水解失效。
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| Sulfo-NHS-Biotin | Sulfo-NHS-Biotin (Sulfosuccinimidyl biotin) is a water soluble biotinylation reagent. |
| NHS-Biotin | NHS-Biotin (Succinimidyl Biotin; Succinimidobiotin) is a primary amine reactive biotinylation reagent. |
| Sulfo-NHS-LC-Biotin | Sulfo-NHS-LC-Biotin, Sulfosuccinimidyl 6-(biotinamido) Hexanoate, is a long chain water soluble biotinylation reagent that is reactive toward primary amine groups. |
| NHS-LC-Biotin | Succinimidyl 6-(biotinamido)hexanoate (NHS-LC-Biotin) is an amino-reactive biotinylation reagent with a long spacer arm. |
| Sulfo-NHS-SS-Biotin | Sulfosuccinimidyl-2-(biotinamido)-ethyl-1,3-dithiopropionate (Sulfo-NHS-SS-Biotin) is a cleavable, water-soluble, amino-reactive biotinylation reagent. |
| NHS-SS-Biotin | NHS-SS-Biotin, Succinimidyl-2-(biotinamido)-ethyl-1,3'-dithiopropionate, is an amine-reactive biotinylation reagent that contains a reducible disulfide. |

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