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抗体药物偶联物 (ADC) 是一种蛋白质—通常为单克隆抗体 (mAb)——通过ADC交联剂共价结合(偶联)到小分子药物。 mAb的定位能力与强效抗癌药物相结合,可敏感地辨析健康细胞和患病细胞。 鉴于偶联药物的效力,开发这些生物治疗药物比单独开发mAb更加困难,包括设计用于详细表征ADC的 UHPLC系统、质谱系统和LC色谱柱,能让您更方便地分离和表征这些新型分子。
ADC药物的药效和清除率都与药物抗体偶联比(DAR)值有关,因此在药物开发过程中必须对其精确分析。尺寸排阻色谱法和疏水色谱法是在天然生理条件下检测DAR的两种最常用的方法。

相关资料:
Mouse Anti-vc-PAB-MMAE mAb (B11F11)
Rabbit Anti-MMAF pAb
Mouse Anti-MMAF mAb (F3B11)
Mouse Anti-MMAE / F mAb (B12A2)
Mouse Anti-MMAE /F mAb (C12A1)
Rabbit Anti-DM1/4 pAb
Mouse Anti-DM1/4 mAb (F1D5)
Mouse Anti-DM1/4 mAb (G2F3)
Rabbit Anti-Calicheamicin pAb
Mouse Anti-Calicheamicin mAb (B1G9)
Mouse Anti-Calicheamicin mAb (C1F12)
Rabbit Anti-Duocarmycin pAb
Mouse Anti-Duocarmycin mAb (E11A1)
Mouse Anti-Duocarmycin mAb (H7A9)
Mouse Anti-Duocarmycin mAb (E6B3)
Rabbit Anti-PNU-159682 pAb
Mouse Anti-PNU-159682 mAb (F7F2)
Mouse Anti-PNU-159682 mAb (C1E3)
Mouse Anti-PNU-159682 mAb (D12H11)
Rabbit Anti-Amanitin pAb
Mouse Anti-Amanitin mAb (H3E1)
Mouse Anti-Amanitin mAb (H12D6)
Mouse Anti-Amanitin mAb (C2C4)
Rabbit Anti-SN38 pAb
Mouse Anti-SN38 mAb (10F11A9D6)
Mouse Anti-SN38 mAb (8E10F12F3)
Mouse Anti-SN38 mAb (8E10A4A1)
Rabbit Anti-PBD SG3199 pAb
Mouse Anti-PBD SG3199 (7H6H9A6) mAb
Mouse Anti-PBD SG3199 (8G2H12A9) mAb
Mouse Anti-PBD SG3199 (8B3D12G1) mAb
Dolastatin 10 Cas号:110417-88-4 微管蛋白聚合抑制剂
Monomethyl Dolastatin 10 Cas号:203849-91-6单甲基澳瑞他汀
Auristatin E Cas号:160800-57-7 澳瑞他汀
Monomethyl Auristatin E 474645-27-7微管相关抑制剂
Auristatin F Cas号:163768-50-1 澳瑞他汀
Monomethyl Auristatin F Cas号:745017-94-1
HTI-286 228266-40-8
Tubulysin M 205304-86-5
Maytansinoid AP-3 66547-09-9
Maytansinol 57103-68-1
DM1 139504-50-0
DM4 799840-96-3
Boc-Val-Dil-Dap-OH
Boc-Val-Dil-Dap-Phe-OMe
Boc-Val-Dil-Dap-Doe
Boc-Val-Dil-Dap-Nrp
Boc-N-Me-Val-Val-Dil-Dap-OH
Tubulysin IM-1
Tubulysin IM-2
Tubulysin IM-3
Duocarmycin SA 152785-82-5
Duocarmycin TM
Duocarmycin MA
Duocarmycin DM
Nemorubicin 108852-90-0
PNU-159682 202350-68-3
Calicheamicin g1 108212-75-5
Acetyl-Calicheamicin g1 108212-76-6
a-Amanitin 23109-05-9
PBD-dimer 1222490-34-7
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